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Boost the natural testosterone production. Has anti-estrogenic properties.
Great for post cycle therapy.
Appearance: White capsule shaped tablet with round surface.
Packing: 100 tablets
Clomiphene citrate is in existence since 1960s, during which period it was first used to treat cases of oligomenorrhea. Its next usage was its application to the treatment of anovulation.
Clomiphene citrate is a selective estrogen receptor modulator (SERM) having an affinity to increase the production of gonadotropins by controlling hypothalamus. Mainly it is used in female infertility cases related to ovarian stimulation to reverse oligo ovulation or anovulation like infertility in polycystic ovary syndrome. It is also used for ovarian hyper stimulation being a part of in vitro fertilization process. It inhibits estrogen receptors in hypothalamus resulting into inhibition of negative feedback of estrogen on production of gonadotropin.
Clomiphene citrate stimulates hypothalamic pituitary axis. It is found to be helpful in the treatment of secondary male hypogonadism conditions. For this particular range of treatment, it is considered as a better choice than testosterone replacement therapy (TRT) for convenience purposes. As is in the case of testosterone replacement therapy in which the size of the testes shrinks considerably, it does not happen in case of treatment done by Clomiphene citrate in place of TRT. As is evident, that shrinkage of testes causes decrease in fertility. So that risk is gone with the usage of Clomiphene citrate. TRT can lead a man to sterility.
Clomiphene citrate is generally used by male bodybuilders and athletes who prefer to use anabolic steroids for the purpose of binding the estrogen receptors in their body. This in turn blocks the effects of estrogen like gynecomastia. It also helps in restoration of body's natural production capability of testosterone. Usually it is termed as 'recovery drug' and is taken towards the end of steroid cycle by athletes and bodybuilders. Clomiphene citrate is an anti estrogen for attaining improvement in recovery of natural testosterone producing capacity after a cycle. It is used for improving testosterone production of endurance athletes. It is also effective in reduction of risk of gynecomastia during a cycle having usage of aromatizable steroids.
Clomiphen is a triphenylethylene derivative a far relative of diethylstilbestrol. Clomiphene citrate functions as a selective estrogen receptor modulator. It inhibits estrogen binding to estrogen receptors and has mixed agonist and antagonist activity depending on the target tissue. Commercially clomiphen is available in the market as its dihydrogen citrate salt known as Clomiphene citrate. It consists of two stereoisomers - zu-clomiphen (38%) and en-clomiphen (62%). These two isomers were initially termed as cis-isomer and trans-isomer respectively. Where the en-clomiphen clears off quickly, the zu-clomiphen has a significant longer life. These two isomers have mixes estrogenic and antiestrogenic effects. Zu-clomiphen has higher estrogenic tendency than en-clomiphen.
Clomiphene citrate gets absorbed by the gastrointestinal tract. First 50% excretion of oral dose of clomiphen occurs in fifth day after its intake. However the rest takes almost six weeks. In females it works as a fertility drug and increases the number of eggs released for possible fertilization thereby increasing the chances of a female getting pregnant. It is generally administered to women who are not able to ovulate on regular basis or in those cases where pregnancy has not occurred for long.
|Package||100 tabs x 50 mg = 5000 mg|